Browse Target: Membrane Receptor Category: Small molecule receptor (family A GPCR)

Target ID Target Name Target Organism # Natural Product # Activity Record
NPT4161 G-protein coupled receptor 81 Homo sapiens 2 2
NPT4903 Hydroxycarboxylic acid receptor 2 Rattus norvegicus 1 4
NPT4904 HM74 nicotinic acid GPCR Homo sapiens 1 4
NPT4905 Hydroxycarboxylic acid receptor 2 Mus musculus 1 6
NPT525 Hydroxycarboxylic acid receptor 2 Homo sapiens 19 63
NPT1627 G-protein coupled receptor 35 Homo sapiens 14 54
NPT5097 G protein-coupled receptor GPR35 Rattus norvegicus 1 1
NPT6197 Glucose-dependent insulinotropic receptor Homo sapiens 1 3
NPT6199 Glucose-dependent insulinotropic receptor Mus musculus 1 1
NPT1169 Cannabinoid CB2 receptor Mus musculus 17 21
NPT1170 Cannabinoid CB1 receptor Mus musculus 15 25
NPT1287 Cannabinoid CB2 receptor Homo sapiens 66 202
NPT1361 Cannabinoid CB1 receptor Rattus norvegicus 18 75
NPT1362 Cannabinoid receptor Homo sapiens 2 3
NPT232 Cannabinoid CB1 receptor Homo sapiens 73 222
NPT3955 Cannabinoid CB2 receptor Rattus norvegicus 4 8
NPT4118 Cannabinoid receptor Rattus norvegicus 3 11
NPT5404 Cannabinoid receptor Mus musculus 2 2
NPT6035 Sphingosine 1-phosphate receptor Edg-1 Homo sapiens 1 22
NPT6036 Sphingosine 1-phosphate receptor Edg-3 Homo sapiens 1 17
NPT6037 Sphingosine 1-phosphate receptor Edg-5 Homo sapiens 1 9
NPT6115 Sphingosine 1-phosphate receptor Edg-6 Homo sapiens 1 11
NPT6116 Sphingosine 1-phosphate receptor Edg-8 Homo sapiens 1 11
NPT3731 Free fatty acid receptor 2 Homo sapiens 2 2
NPT4000 Free fatty acid receptor 1 Mus musculus 1 2
NPT4003 G-protein coupled receptor 120 Homo sapiens 2 4
NPT869 Free fatty acid receptor 1 Homo sapiens 6 16
NPT256 Cysteinyl leukotriene receptor 1 Homo sapiens 1 6
NPT3068 Leukotriene B4 receptor 1 Homo sapiens 5 19
NPT3069 Leukotriene B4 receptor Homo sapiens 1 4
NPT4030 Oxoeicosanoid receptor 1 Homo sapiens 5 7
NPT4528 Cysteinyl leukotriene receptor 1 Cavia porcellus 1 1
NPT4120 G-protein coupled receptor 55 Homo sapiens 13 18
NPT1372 Platelet activating factor receptor Cavia porcellus 10 26
NPT274 Platelet activating factor receptor Homo sapiens 4 5
NPT1011 Prostanoid EP1 receptor Mus musculus 2 6
NPT1012 Prostanoid EP2 receptor Mus musculus 2 7
NPT1013 Prostanoid EP3 receptor Mus musculus 2 6
NPT1014 Prostanoid EP4 receptor Mus musculus 2 9
NPT1015 Prostanoid IP receptor Homo sapiens 3 11
NPT1030 Prostanoid EP1 receptor Rattus norvegicus 1 1
NPT2763 Prostanoid FP receptor Bos taurus 1 3
NPT2764 Prostanoid FP receptor Homo sapiens 2 8
NPT2765 Prostanoid EP1 receptor Homo sapiens 2 8
NPT2766 Prostanoid EP2 receptor Homo sapiens 3 16
NPT2767 Prostanoid EP3 receptor Homo sapiens 2 8
NPT2768 Prostanoid EP4 receptor Homo sapiens 2 19
NPT2769 Thromboxane A2 receptor Homo sapiens 1 3
NPT2770 Prostanoid DP receptor Homo sapiens 1 2
NPT2772 Prostanoid FP receptor Mus musculus 1 3
NPT4331 Prostanoid EP2 receptor Rattus norvegicus 1 3
NPT4332 Prostanoid EP4 receptor Rattus norvegicus 1 3
NPT3037 G-protein coupled estrogen receptor 1 Homo sapiens 1 10
NPT3948 G-protein coupled bile acid receptor 1 Mus musculus 2 2
NPT745 G-protein coupled bile acid receptor 1 Homo sapiens 52 85
NPT1295 Muscarinic acetylcholine receptor M1 Mus musculus 2 7
NPT1296 Muscarinic acetylcholine receptor M2 Mus musculus 3 7
NPT1297 Muscarinic acetylcholine receptor M3 Mus musculus 1 2
NPT1299 Muscarinic acetylcholine receptors; M2 & M3 Homo sapiens 2 2
NPT1300 Muscarinic acetylcholine receptors; M1 & M2 Homo sapiens 2 3
NPT1301 Muscarinic acetylcholine receptor M2 Rattus norvegicus 7 21
NPT1302 Muscarinic acetylcholine receptor Homo sapiens 8 26
NPT1303 Muscarinic acetylcholine receptor M3 Rattus norvegicus 6 10
NPT262 Muscarinic acetylcholine receptor M1 Homo sapiens 20 74
NPT263 Muscarinic acetylcholine receptor M2 Homo sapiens 17 59
NPT264 Muscarinic acetylcholine receptor M3 Homo sapiens 23 48
NPT265 Muscarinic acetylcholine receptor M4 Homo sapiens 11 34
NPT266 Muscarinic acetylcholine receptor M5 Homo sapiens 16 41
NPT2843 Muscarinic acetylcholine receptor M2 Sus scrofa 2 2
NPT3977 Muscarinic acetylcholine receptor M5 Rattus norvegicus 2 2
NPT420 Muscarinic acetylcholine receptor M3 Cavia porcellus 1 5
NPT422 Muscarinic acetylcholine receptor Rattus norvegicus 7 81
NPT432 Muscarinic acetylcholine receptor M4 Rattus norvegicus 5 8
NPT5996 Muscarinic receptor M1 and M2 Rattus norvegicus 1 1
NPT5997 Muscarinic acetylcholine receptor M1 Bos taurus 1 2
NPT6000 Muscarinic acetylcholine receptor Mus musculus 1 1
NPT6202 Muscarinic acetylcholine receptor DM1 Drosophila melanogaster 1 4
NPT95 Muscarinic acetylcholine receptor M1 Rattus norvegicus 96 171
NPT1386 Adrenergic receptor beta Homo sapiens 14 29
NPT1788 Alpha-1a adrenergic receptor Homo sapiens 18 39
NPT1789 Alpha-1b adrenergic receptor Homo sapiens 14 26
NPT219 Alpha-1a adrenergic receptor Rattus norvegicus 21 43
NPT220 Alpha-1b adrenergic receptor Rattus norvegicus 19 32
NPT221 Alpha-1d adrenergic receptor Homo sapiens 15 37
NPT222 Alpha-2a adrenergic receptor Homo sapiens 29 69
NPT223 Alpha-2b adrenergic receptor Homo sapiens 24 47
NPT224 Alpha-2c adrenergic receptor Homo sapiens 24 49
NPT225 Beta-1 adrenergic receptor Homo sapiens 7 37
NPT226 Beta-2 adrenergic receptor Homo sapiens 32 66
NPT227 Beta-3 adrenergic receptor Homo sapiens 8 19
NPT2838 Beta-1 adrenergic receptor Sus scrofa 2 2
NPT2839 Beta-2 adrenergic receptor Sus scrofa 2 2
NPT2840 Adrenergic receptor alpha Homo sapiens 2 2
NPT3048 Alpha-1d adrenergic receptor Rattus norvegicus 10 16
NPT3049 Alpha-2a adrenergic receptor Sus scrofa 1 1
NPT3050 Alpha-2 adrenergic receptor Mus musculus 2 7
NPT3051 Alpha-1a adrenergic receptor Bos taurus 5 9
NPT3057 Alpha-2a adrenergic receptor Bos taurus 2 4
NPT3059 Alpha-2b adrenergic receptor Rattus norvegicus 4 6
NPT4333 Adrenergic receptor beta Rattus norvegicus 9 27
NPT4554 Alpha-1b adrenergic receptor Mesocricetus auratus 5 6
NPT4555 Adrenergic receptors; alpha-1 A & B Homo sapiens 1 2
NPT4557 Adrenergic receptor beta; ADRB1 & ADRB3 Homo sapiens 1 1
NPT4558 Beta-1 adrenergic receptor Rattus norvegicus 7 39
NPT4630 Beta-2 adrenergic receptor Bos taurus 3 5
NPT4632 Beta-2 adrenergic receptor Rattus norvegicus 3 3
NPT4663 Beta-2 adrenergic receptor Canis lupus familiaris 6 14
NPT4893 Alpha-1a adrenergic receptor Oryctolagus cuniculus 2 2
NPT4894 Alpha-2a adrenergic receptor Rattus norvegicus 1 1
NPT4913 Beta-1 adrenergic receptor Cavia porcellus 5 37
NPT4914 Beta-2 adrenergic receptor Cavia porcellus 5 25
NPT4915 Beta-3 adrenergic receptor Rattus norvegicus 1 2
NPT5860 Adrenergic receptor beta; ADRB1 & ADRB2 Homo sapiens 3 10
NPT968 Adrenergic receptor alpha-1 Rattus norvegicus 17 70
NPT969 Adrenergic receptor alpha-2 Rattus norvegicus 18 108
NPT970 Adrenergic receptor alpha-1 Homo sapiens 8 13
NPT971 Adrenergic receptor alpha-2 Homo sapiens 7 44
NPT972 Adrenergic receptor alpha Rattus norvegicus 7 10
NPT1786 Dopamine receptor Homo sapiens 4 4
NPT1811 Dopamine D5 receptor Homo sapiens 8 9
NPT1857 Dopamine D1 receptor Rattus norvegicus 31 55
NPT1858 Dopamine D2 receptor Rattus norvegicus 33 83
NPT242 Dopamine D1 receptor Homo sapiens 103 211
NPT243 Dopamine D2 receptor Homo sapiens 49 164
NPT244 Dopamine D3 receptor Homo sapiens 23 77
NPT245 Dopamine D4 receptor Homo sapiens 11 24
NPT3052 Dopamine receptor Rattus norvegicus 3 5
NPT3056 Dopamine D3 receptor Rattus norvegicus 7 11
NPT3471 Dopamine D2 receptor Bos taurus 4 29
NPT4411 Dopamine receptors; D2 & D4 Homo sapiens 4 4
NPT4657 Dopamine D1 receptor Bos taurus 1 8
NPT4659 Dopamine receptor Bos taurus 1 7
NPT4661 Dopamine D4 receptor Rattus norvegicus 1 3
NPT4666 Dopamine receptor D2 and D3 Rattus norvegicus 1 2
NPT5857 Dopamine D1 receptor Mus musculus 2 2
NPT251 Histamine H1 receptor Homo sapiens 14 47
NPT252 Histamine H2 receptor Homo sapiens 8 26
NPT3936 Histamine H4 receptor Rattus norvegicus 3 5
NPT4288 Histamine H1 receptor Cavia porcellus 9 35
NPT4289 Histamine H2 receptor Cavia porcellus 5 18
NPT4290 Histamine H2 receptor Rattus norvegicus 1 1
NPT4292 Histamine H1 receptor Mus musculus 1 2
NPT4293 Histamine H1 receptor Rattus norvegicus 5 8
NPT4294 Histamine H3 receptor Mus musculus 1 1
NPT4295 Histamine H4 receptor Mus musculus 1 4
NPT4297 Histamine H4 receptor Cavia porcellus 1 1
NPT986 Histamine H3 receptor Rattus norvegicus 9 16
NPT987 Histamine H3 receptor Homo sapiens 7 38
NPT988 Histamine H4 receptor Homo sapiens 5 39
NPT989 Histamine H3 receptor Cavia porcellus 5 9
NPT1776 Serotonin 1 (5-HT1) receptor Rattus norvegicus 15 22
NPT1777 Serotonin 2 (5-HT2) receptor Rattus norvegicus 19 52
NPT1778 Serotonin 2a (5-HT2a) receptor Rattus norvegicus 21 47
NPT1779 Serotonin 2b (5-HT2b) receptor Rattus norvegicus 11 13
NPT1784 Serotonin 5a (5-HT5a) receptor Homo sapiens 17 32
NPT1785 Serotonin 7 (5-HT7) receptor Homo sapiens 42 67
NPT2695 Serotonin 2a (5-HT2a) receptor Mus musculus 2 2
NPT2776 Serotonin 1e (5-HT1e) receptor Homo sapiens 7 10
NPT288 Serotonin 1a (5-HT1a) receptor Rattus norvegicus 28 77
NPT289 Serotonin 1b (5-HT1b) receptor Rattus norvegicus 15 39
NPT290 Serotonin 2a (5-HT2a) receptor Homo sapiens 52 118
NPT291 Serotonin 2b (5-HT2b) receptor Homo sapiens 47 95
NPT292 Serotonin 2c (5-HT2c) receptor Homo sapiens 48 117
NPT293 Serotonin 4 (5-HT4) receptor Cavia porcellus 8 24
NPT294 Serotonin 6 (5-HT6) receptor Homo sapiens 24 61
NPT2958 Serotonin 4 (5-HT4) receptor Rattus norvegicus 2 9
NPT3053 Serotonin 2c (5-HT2c) receptor Mus musculus 1 1
NPT3055 Serotonin receptor (2b and 2c) Homo sapiens 1 1
NPT4011 Serotonin 4 (5-HT4) receptor Homo sapiens 4 21
NPT4041 Serotonin 7 (5-HT7) receptor Rattus norvegicus 5 8
NPT4043 Serotonin 2 (5-HT2) receptor Homo sapiens 2 4
NPT4045 Serotonin (5-HT) receptor Homo sapiens 1 1
NPT438 Serotonin 2c (5-HT2c) receptor Rattus norvegicus 14 23
NPT4579 Serotonin 1d (5-HT1d) receptor Sus scrofa 2 4
NPT5249 Serotonin 5a (5-HT5a) receptor Mus musculus 1 1
NPT5250 Serotonin receptor 2a and 2c (5HT2A and 5HT2C) Rattus norvegicus 1 3
NPT5251 Serotonin 1d (5-HT1d) receptor Rattus norvegicus 1 2
NPT5254 Serotonin 2 (5-HT2) receptor Mus musculus 1 2
NPT5255 Serotonin 1a (5-HT1a) receptor Mus musculus 2 2
NPT5256 Serotonin 1f (5-HT1f) receptor Homo sapiens 1 1
NPT5856 Serotonin 2a (5-HT2a) receptor Bos taurus 1 1
NPT92 Serotonin 1a (5-HT1a) receptor Homo sapiens 63 137
NPT973 Serotonin 1b (5-HT1b) receptor Homo sapiens 14 37
NPT974 Serotonin 1d (5-HT1d) receptor Homo sapiens 14 32
NPT4319 Trace amine-associated receptor 1 Macaca mulatta 2 2
NPT4320 Trace amine-associated receptor 1 Rattus norvegicus 4 11
NPT4321 Trace amine-associated receptor 1 Mus musculus 4 10
NPT976 Trace amine-associated receptor 1 Homo sapiens 12 25
NPT4046 Melatonin receptor 1A Homo sapiens 4 71
NPT4047 Melatonin receptor 1B Homo sapiens 4 62
NPT4906 Melatonin receptor Gallus gallus 4 19
NPT5862 Melatonin receptor Homo sapiens 1 28
NPT5863 Melatonin receptor 1B Gallus gallus 1 1
NPT5866 Melatonin receptor 1C Xenopus laevis 1 2
NPT1315 Adenosine A1 receptor Rattus norvegicus 69 198
NPT1316 Adenosine A2a receptor Rattus norvegicus 33 70
NPT1760 Adenosine A3 receptor Rattus norvegicus 8 16
NPT216 Adenosine A1 receptor Homo sapiens 20 64
NPT217 Adenosine A2a receptor Homo sapiens 19 75
NPT218 Adenosine A3 receptor Homo sapiens 44 102
NPT2554 Adenosine A2 receptor Rattus norvegicus 17 62
NPT2555 Adenosine receptors; A1 & A3 Rattus norvegicus 15 15
NPT2687 Adenosine receptor A2a and A3 Rattus norvegicus 4 4
NPT2812 Adenosine A2 receptor Homo sapiens 7 12
NPT3054 Adenosine A2b receptor Rattus norvegicus 3 6
NPT4059 Adenosine A2b receptor Homo sapiens 10 36
NPT4262 Adenosine A2a receptor Cavia porcellus 5 11
NPT4749 Adenosine receptors; A1 & A2 Rattus norvegicus 5 15
NPT4757 Adenosine receptors; A1 & A2 Homo sapiens 5 6
NPT5049 Adenosine A1 receptor Bos taurus 4 18
NPT5443 Adenosine receptors; A1 & A2a Rattus norvegicus 1 1
NPT5444 Adenosine receptor Rattus norvegicus 3 15
NPT5445 Adenosine A2b receptor Mus musculus 2 2
NPT5448 Adenosine receptors; A1 & A3 Homo sapiens 1 2
NPT1391 Pyrimidinergic receptor P2Y6 Homo sapiens 10 39
NPT2757 Purinergic receptor P2Y12 Homo sapiens 13 24
NPT3825 Purinergic receptor P2Y1 Homo sapiens 8 18
NPT3826 Purinergic receptor P2Y2 Homo sapiens 14 102
NPT3827 Pyrimidinergic receptor P2Y4 Homo sapiens 7 24
NPT3828 Pyrimidinergic receptor P2Y4 Rattus norvegicus 3 3
NPT3829 Purinergic receptor P2Y11 Homo sapiens 6 11
NPT3831 Purinergic receptor P2Y1 Rattus norvegicus 3 4
NPT3832 Purinergic receptor P2Y2 Rattus norvegicus 1 1
NPT3833 Purinergic receptor P2Y2 Mus musculus 1 3
NPT4492 P2Y purinoceptor 1 Meleagris gallopavo 5 13
NPT4493 Purinergic receptor P2Y12 Rattus norvegicus 2 2
NPT4712 Purinergic receptor P2Y14 Homo sapiens 4 12
NPT4962 Pyrimidinergic receptor P2Y6 Rattus norvegicus 1 2